BIOPEP-UWM: Report

ID 10132
Name ACE inhibitor
sequence
LMP

Function:
Inhibitor of Angiotensin-Converting Enzyme (ACE) (EC 3.4.15.1) (MEROPS ID: M02-001)
 
Number of residues
3
Activity code
ah
Activity :
ACE inhibitor
Chemical mass 359.4841 Monoisotopic mass 359.1872
IC50 :
15.80 µM



Bibliographic data:
Authors
Lammi C., Boschin G., Bollati C., Arnoldi A., Galaverna G., Dellafiora L.
Title
A heuristic, computer-driven and top-down approach to identify novel bioactive peptides: a proof-of-principle on angiotensin I converting enzyme inhibitory peptides. Food Res. Int., 150 A, 110753, 2021
Year Source
2021 Journal



Additional information:
BIOPEP-UWM database of bioactive peptides


SMILES: N[C@@]([H])(CC(C)C)C(=O)N[C@@]([H])(CCSC)C(=O)N1[C@@]([H])(CCC1)C(=O)O

InChI=1S/C16H29N3O4S/c1-10(2)9-11(17)14(20)18-12(6-8-24-3)15(21)19-7-4-5-13(19)16(22)23/h10-13H,4-9,17H2,1-3H3,(H,18,20)(H,22,23)/t11-,12-,13-/m0/s1

InChIKey=GNRPTBRHRRZCMA-AVGNSLFASA-N


Information concerning Angiotensin-Converting Enzyme (ACE) is available in MEROPS database of proteolytic enzymes (http://merops.sanger.ac.uk/); ID: M02-001


IC50 measured using cel-based assay; 6.8 µM
Lammi C., Boschin G., Bollati C., Arnoldi A., Galaverna G., Dellafiora L., 2021, A heuristic, computer-driven and top-down approach to identify novel bioactive peptides: a proof-of-principle on angiotensin I converting enzyme inhibitory peptides. Food Res. Int., 150 A, 110753



Database reference: