BIOPEP-UWM: Report

ID 10485
Name Acetylcholinesterase inhibitor
sequence
SQSQ

Function:
Inhibitor of Acetylcholinesterase (EC 3.1.1.7)
 
Number of residues
4
Activity code
ache
Activity :
AChE inhibitor
Chemical mass 448.4272 Monoisotopic mass 448.1911
IC50 :
15488.00 µM



Bibliographic data:
Authors
Asen N.D., Okagu O.D., Udenigwe C.C., Aluko R.E.
Title
In vitro inhibition of acetylcholinesterase activity by yellow field pea (Pisum sativum) protein-derived peptides as revealed by kinetics and molecular docking. Front. Nutr., 9, 2022
Year Source
2022 Journal



Additional information:
BIOPEP-UWM database of bioactive peptides


SMILES: N[C@@]([H])(CO)C(=O)N[C@@]([H])(CCC(=O)N)C(=O)N[C@@]([H])(CO)C(=O)N[C@@]([H])(CCC(=O)N)C(=O)O

InChI=1S/C16H28N6O9/c17-7(5-23)13(27)20-8(1-3-11(18)25)14(28)22-10(6-24)15(29)21-9(16(30)31)2-4-12(19)26/h7-10,23-24H,1-6,17H2,(H2,18,25)(H2,19,26)(H,20,27)(H,21,29)(H,22,28)(H,30,31)/t7-,8-,9-,10-/m0/s1

InChIKey=VSWOVIIPXAMIHU-XKNYDFJKSA-N

The IC50 value was calculated in μmol/L.



Database reference: