BIOPEP-UWM: Report

ID 10489
Name Acetylcholinesterase inhibitor
sequence
RSQSQ

Function:
Inhibitor of Acetylcholinesterase (EC 3.1.1.7)
 
Number of residues
5
Activity code
ache
Activity :
AChE inhibitor
Chemical mass 604.6124 Monoisotopic mass 604.2920
IC50 :
1122.00 µM



Bibliographic data:
Authors
Asen N.D., Okagu O.D., Udenigwe C.C., Aluko R.E.
Title
In vitro inhibition of acetylcholinesterase activity by yellow field pea (Pisum sativum) protein-derived peptides as revealed by kinetics and molecular docking. Front. Nutr., 9, 2022
Year Source
2022 Journal



Additional information:
BIOPEP-UWM database of bioactive peptides


SMILES: N[C@@]([H])(CCCNC(=N)N)C(=O)N[C@@]([H])(CO)C(=O)N[C@@]([H])(CCC(=O)N)C(=O)N[C@@]([H])(CO)C(=O)N[C@@]([H])(CCC(=O)N)C(=O)O

InChI=1S/C22H40N10O10/c23-10(2-1-7-28-22(26)27)17(37)31-13(8-33)19(39)29-11(3-5-15(24)35)18(38)32-14(9-34)20(40)30-12(21(41)42)4-6-16(25)36/h10-14,33-34H,1-9,23H2,(H2,24,35)(H2,25,36)(H,29,39)(H,30,40)(H,31,37)(H,32,38)(H,41,42)(H4,26,27,28)/t10-,11-,12-,13-,14-/m0/s1

InChIKey=FSXVTGQUNXGDLJ-PEDHHIEDSA-N

The IC50 value was calculated in μmol/L.





Database reference: