BIOPEP-UWM: Report

ID 10491
Name Acetylcholinesterase inhibitor
sequence
ETRSQ

Function:
Inhibitor of Acetylcholinesterase (EC 3.1.1.7)
 
Number of residues
5
Activity code
ache
Activity :
AChE inhibitor
Chemical mass 619.6237 Monoisotopic mass 619.2916
IC50 :
912.00 µM



Bibliographic data:
Authors
Asen N.D., Okagu O.D., Udenigwe C.C., Aluko R.E.
Title
In vitro inhibition of acetylcholinesterase activity by yellow field pea (Pisum sativum) protein-derived peptides as revealed by kinetics and molecular docking. Front. Nutr., 9, 2022
Year Source
2022 Journal



Additional information:
BIOPEP-UWM database of bioactive peptides


SMILES: N[C@@]([H])(CCC(=O)O)C(=O)N[C@@]([H])([C@]([H])(O)C)C(=O)N[C@@]([H])(CCCNC(=N)N)C(=O)N[C@@]([H])(CO)C(=O)N[C@@]([H])(CCC(=O)N)C(=O)O

InChI=1S/C23H41N9O11/c1-10(34)17(32-18(38)11(24)4-7-16(36)37)21(41)29-12(3-2-8-28-23(26)27)19(39)31-14(9-33)20(40)30-13(22(42)43)5-6-15(25)35/h10-14,17,33-34H,2-9,24H2,1H3,(H2,25,35)(H,29,41)(H,30,40)(H,31,39)(H,32,38)(H,36,37)(H,42,43)(H4,26,27,28)/t10-,11+,12+,13+,14+,17+/m1/s1

InChIKey=UBLCEYAHFHDAGS-UFRCXNNCSA-N

The IC50 value was calculated in μmol/L.






Database reference: