BIOPEP-UWM: Report
| ID | 10668 |
| Name | Inhibitor of tripeptidyl peptidase II |
| sequence |
| Function: | |||
| Inhibitor of tripeptidyl peptidase II (EC 3.4.14.10) (MEROPS ID: S08.090) | |||
| Number of residues | 2 |
Activity code | tpp2 |
| Activity : | inhibitor of tripeptidyl peptidase II |
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| Chemical mass | 244.3296 | Monoisotopic mass | 244.1781 | |
| IC50 : | 0.00 µM |
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| Bibliographic data: | |
| Authors | |
| Ganellin C. R., Bishop P. B., Bambal R. B., Chan S. M., Law J. K., Marabout B., Luthra P. M., Moore A. N., Peschard O., Bourgeat P., Rose C., Vargas F. | |
| Title | |
| Inhibitors of tripeptidyl peptidase II. 2. Generation of the first novel lead inhibitor of cholecystokinin-8-inactivating peptidase: a strategy for the design of peptidase inhibitors. J. Med. Chem., 43, 664-674, 2000 | |
| Year | Source |
| 2000 | Journal |
| Additional information: |
| BIOPEP-UWM database of bioactive peptides SMILES: N[C@@H](CCCC)C(=O)N[C@@H](CCCC)C(=O)O InChI=1S/C12H24N2O3/c1-3-5-7-9(13)11(15)14-10(12(16)17)8-6-4-2/h9-10H,3-8,13H2,1-2H3,(H,14,15)(H,16,17)/t9-,10-/m0/s1 InChIKey=YWCWRUFTSHXXCO-UWVGGRQHSA-N {Nle} - Norleucine (ID 231 in the BIOPEP-UWM repository of amino acids and modifications) |
| Database reference: |
| BRENDA: Ligand Nle-Nle-OH CAS: Registry No 114148-92-4 ChEMBL: ID CHEMBL2371256 ChemSpider: ID 30846645 EPA CompTox: ID DTXSID60719368 PubChem: CID 56972312 Wikidata: ID Q82657685 |