BIOPEP-UWM: Report

ID 10671
Name Antiviral peptide
sequence
IAEK

Function:
Inhibitor of SARS-CoV-2 parent protease (EC 3.4.22.69) (MEROPS ID: C30.007)
 
Number of residues
4
Activity code
avi
Activity :
antiviral
Chemical mass 459.5356 Monoisotopic mass 459.2684
EC50 :
0.00 µM



Bibliographic data:
Authors
Gambacorta N., Caputo L., Quintieri L., Monaci L., Ciriaco F., Nicolotti O.
Title
Rational discovery of antiviral whey protein-derived small peptides targeting the SARS-CoV-2 main protease. Biomedicines, 10, 1067, 2022
Year Source
2022 Journal



Additional information:
BIOPEP-UWM database of bioactive peptides


SMILES: N[C@@]([H])([C@]([H])(CC)C)C(=O)N[C@@]([H])(C)C(=O)N[C@@]([H])(CCC(=O)O)C(=O)N[C@@]([H])(CCCCN)C(=O)O

InChI=1S/C20H37N5O7/c1-4-11(2)16(22)19(30)23-12(3)17(28)24-13(8-9-15(26)27)18(29)25-14(20(31)32)7-5-6-10-21/h11-14,16H,4-10,21-22H2,1-3H3,(H,23,30)(H,24,28)(H,25,29)(H,26,27)(H,31,32)/t11-,12-,13-,14-,16-/m0/s1

InChIKey=KHPMTTPEKURSEX-YGJAXBLXSA-N




Database reference:
ChemSpider: ID 8429165

PubChem: CID 10253679