BIOPEP-UWM: Report

ID 10814
Name ACE inhibitor
sequence
LGAVPPRY

Function:
Inhibitor of Angiotensin-converting enzyme (EC 3.4.15.1) (MEROPS ID: M02-001)
 
Number of residues
8
Activity code
ah
Activity :
ACE inhibitor
Chemical mass 872.0199 Monoisotopic mass 871.4901
IC50 :
29.30 µM



Bibliographic data:
Authors
Suleman D. N., Sutopo C. C. Y., Hsu J.-L.
Title
Characterization of novel angiotensin-I converting enzyme inhibitory peptides derived from Taiwan red quinoa (Chenopodium formosanum Koidz.) seed proteins using two sequential bioassay guided fractionations. Med. Chem. Res., 33, 107–116, 2024
Year Source
2024 Journal



Additional information:
BIOPEP-UWM database of bioactive peptides


SMILES: N[C@@]([H])(CC(C)C)C(=O)NCC(=O)N[C@@]([H])(C)C(=O)N[C@@]([H])(C(C)C)C(=O)N1[C@@]([H])(CCC1)C(=O)N1[C@@]([H])(CCC1)C(=O)N[C@@]([H])(CCCNC(=N)N)C(=O)N[C@@H](CC1=CC=C(C=C1)O)C(=O)O

InChI=1S/C41H65N11O10/c1-22(2)19-27(42)35(56)46-21-32(54)47-24(5)34(55)50-33(23(3)4)39(60)52-18-8-11-31(52)38(59)51-17-7-10-30(51)37(58)48-28(9-6-16-45-41(43)44)36(57)49-29(40(61)62)20-25-12-14-26(53)15-13-25/h12-15,22-24,27-31,33,53H,6-11,16-21,42H2,1-5H3,(H,46,56)(H,47,54)(H,48,58)(H,49,57)(H,50,55)(H,61,62)(H4,43,44,45)/t24-,27-,28-,29-,30-,31-,33-/m0/s1

InChIKey=ZAFJOXKRKCSDCW-YHAIKQLXSA-N




Database reference: