BIOPEP-UWM: Report
| ID | 2878 |
| Name | Leu-enkephalin-Arg |
| sequence |
| Function: | |||
| Opioid | |||
| Number of residues | 6 |
Activity code | op |
| Activity : | opioid |
|||
| Chemical mass | 711.8064 | Monoisotopic mass | 711.3693 | |
| EC50 : | 0.00 µM |
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| Bibliographic data: | |
| Authors | |
| Schlechtingen G., DeHaven R. N., Daubert J. D., Cassel J. A., Chung N. N., Schiller P. W., Taulane J. P., Goodman M. | |
| Title | |
| Structure-activity relationships of dynorphin a analogues modified in the address sequence. J. Med. Chem., 46, 2104-2109, 2003 | |
| Year | Source |
| 2003 | Journal |
| Additional information: |
| BIOPEP-UWM database of bioactive peptides SMILES: [H][C@](N)(Cc1ccc(O)cc1)C(=O)NCC(=O)NCC(=O)N[C@@]([H])(Cc1ccccc1)C(=O)N[C@@]([H])(CC(C)C)C(=O)N[C@@]([H])(CCCNC(N)=N)C(O)=O InChI=1S/C34H49N9O8/c1-20(2)15-26(31(48)42-25(33(50)51)9-6-14-38-34(36)37)43-32(49)27(17-21-7-4-3-5-8-21)41-29(46)19-39-28(45)18-40-30(47)24(35)16-22-10-12-23(44)13-11-22/h3-5,7-8,10-13,20,24-27,44H,6,9,14-19,35H2,1-2H3,(H,39,45)(H,40,47)(H,41,46)(H,42,48)(H,43,49)(H,50,51)(H4,36,37,38)/t24-,25-,26-,27-/m0/s1 InChIKey=ILBHHEXPXBRSKB-FWEHEUNISA-N Inhibitor of Carboxypeptidase E (EC 3.4.17.10) (MEROPS ID: M20.001) according to the BRENDA database |
| Database reference: |
| ACToR: ID 75106-70-6 BindingDB: ID 50128084 BRENDA: Ligand Tyr-Gly-Gly-Phe-Leu-Arg ChEMBL: ID CHEMBL63188 ChemIDplus: ID 075106706, 082008604 ChemSpider: ID 108826 FDA SRS: ID V1PIQ8ZW62 J-GLOBAL: ID 200907011131312603 Nikkaji: ID J293.206G PepBank: Peptide YGGFLR PubChem: CID 121999 ZINC: ID ZINC000026187176 |