BIOPEP-UWM: Report

ID 8350
Name ACE inhibitor from cuttlefish (Sepia officinalis)
sequence
KNGDGY

Function:
Inhibitor of Angiotensin-Converting Enzyme (ACE) (EC 3.4.15.1) (MEROPS ID: M02-001)
 
Number of residues
6
Activity code
ah
Activity :
ACE inhibitor
Chemical mass 652.6519 Monoisotopic mass 652.2807
IC50 :
51.63 µM



Bibliographic data:
Authors
Balti R., Bougatef A., Sila A., Guillochon D., Dhulster P., Nedjar-Arroume N.
Title
Nine novel angiotensin I-converting enzyme (ACE) inhibitory peptides from cuttlefish (Sepia officinalis) muscle protein hydrolysates and antihypertensive effect of the potent active peptide in spontaneously hypertensive rats. Food Chem., 170, 519-525
Year Source
2015 Journal



Additional information:
BIOPEP-UWM database of bioactive peptides


SMILES: N[C@@]([H])(CCCCN)C(=O)N[C@@]([H])(CC(=O)N)C(=O)NCC(=O)N[C@@]([H])(CC(=O)O)C(=O)NCC(=O)N[C@@]([H])(Cc1ccc(O)cc1)C(=O)O

InChI=1S/C27H40N8O11/c28-8-2-1-3-16(29)24(42)35-17(10-20(30)37)25(43)31-12-21(38)33-18(11-23(40)41)26(44)32-13-22(39)34-19(27(45)46)9-14-4-6-15(36)7-5-14/h4-7,16-19,36H,1-3,8-13,28-29H2,(H2,30,37)(H,31,43)(H,32,44)(H,33,38)(H,34,39)(H,35,42)(H,40,41)(H,45,46)/t16-,17-,18-,19-/m0/s1

InChIKey=KUYGHLBJQIXGRH-VJANTYMQSA-N



Database reference:
EROP-Moscow: ID E21351

FeptideDB: ID 8350