BIOPEP-UWM: Report

ID 8351
Name ACE inhibitor from cuttlefish (Sepia officinalis)
sequence
STHGVY

Function:
Inhibitor of Angiotensin-Converting Enzyme (ACE) (EC 3.4.15.1) (MEROPS ID: M02-001)
 
Number of residues
6
Activity code
ah
Activity :
ACE inhibitor
Chemical mass 662.6897 Monoisotopic mass 662.3014
IC50 :
19.30 µM



Bibliographic data:
Authors
Balti R., Bougatef A., Sila A., Guillochon D., Dhulster P., Nedjar-Arroume N.
Title
Nine novel angiotensin I-converting enzyme (ACE) inhibitory peptides from cuttlefish (Sepia officinalis) muscle protein hydrolysates and antihypertensive effect of the potent active peptide in spontaneously hypertensive rats. Food Chem., 170, 519-525
Year Source
2015 Journal



Additional information:
BIOPEP-UWM database of bioactive peptides


SMILES: N[C@@H](CO)C(=O)N[C@@H]([C@H](O)C)C(=O)N[C@@H](CC1=C[N]([H])C=N1)C(=O)NCC(=O)N[C@@H](C(C)C)C(=O)N[C@@H](CC2=CC=C(C=C2)O)C(=O)O

InChI=1S/C29H42N8O10/c1-14(2)23(27(44)35-21(29(46)47)8-16-4-6-18(40)7-5-16)36-22(41)11-32-26(43)20(9-17-10-31-13-33-17)34-28(45)24(15(3)39)37-25(42)19(30)12-38/h4-7,10,13-15,19-21,23-24,38-40H,8-9,11-12,30H2,1-3H3,(H,31,33)(H,32,43)(H,34,45)(H,35,44)(H,36,41)(H,37,42)(H,46,47)/t15-,19+,20+,21+,23+,24+/m1/s1

InChIKey=VLLDORWGGVRVNR-NRWKVABUSA-N



Database reference:
FeptideDB: ID 8351