BIOPEP-UWM: Report

ID 8438
Name ACE inhibitor
sequence
FCVLRP

Function:
Inhibitor of Angiotensin-Converting Enzyme (ACE) (EC 3.4.15.1) (MEROPS ID: M02-001)
 
Number of residues
6
Activity code
ah
Activity :
ACE inhibitor
Chemical mass 733.9205 Monoisotopic mass 733.3933
IC50 :
12.30 µM



Bibliographic data:
Authors
He H.-L., Chen X.-L., Sun C.-Y., Zhang Y.-Z., Zhou B.-C.
Title
Analysis of novel angiotensin-I-converting enzyme inhibitory peptides from protease-hydrolyzed marine shrimp Acetes chinensis. J. Peptide Sci., 12, 726-733, 2006
Year Source
2006 Journal



Additional information:
BIOPEP database of bioactive peptides


SMILES: N[C@@]([H])(Cc1ccccc1)C(=O)N[C@@]([H])(CS)C(=O)N[C@@]([H])(C(C)C)C(=O)N[C@@]([H])(CC(C)C)C(=O)N[C@@]([H])(CCCNC(=N)N)C(=O)N1[C@@]([H])(CCC1)C(=O)O

InChI=1S/C34H55N9O7S/c1-19(2)16-24(29(45)39-23(12-8-14-38-34(36)37)32(48)43-15-9-13-26(43)33(49)50)40-31(47)27(20(3)4)42-30(46)25(18-51)41-28(44)22(35)17-21-10-6-5-7-11-21/h5-7,10-11,19-20,22-27,51H,8-9,12-18,35H2,1-4H3,(H,39,45)(H,40,47)(H,41,44)(H,42,46)(H,49,50)(H4,36,37,38)/t22-,23-,24-,25-,26-,27-/m0/s1

InChIKey: QIJYKMFKXJOOGS-QCOJBMJGSA-N


Information concerning Angiotensin-Converting Enzyme (ACE) is available in MEROPS database of proteolytic enzymes (http://merops.sanger.ac.uk/); ID: M02-001



Database reference:
AHTPDB: ID 1039, 5352, 6196

EROP-Moscow: ID E07060

SATPdb: ID satpdb23192