BIOPEP-UWM: Report

ID 9002
Name ACE inhibitor from thornback ray muscle (Raja clavata)
sequence
ESAGIH

Function:
Inhibitor of Angiotensin-Converting Enzyme (ACE) (EC 3.4.15.1) (MEROPS ID: M02-001)
 
Number of residues
6
Activity code
ah
Activity :
ACE inhibitor
Chemical mass 612.6311 Monoisotopic mass 612.2858
IC50 :
371.60 µM



Bibliographic data:
Authors
Lassoued I., Mora L., Barkia, Aristoy M.-C., Nasri M., Toldra F.
Title
Angiotensin I-converting enzyme inhibitory peptides FQPSF and LKYPI identified in Bacillus subtilis A26 hydrolysate of thornback ray muscle. Int. J. Food Sci. Food Technol., 51, 1604-1609, 2016
Year Source
2016 Journal



Additional information:
BIOPEP-UWM database of bioactive peptides


SMILES: N[C@@H](CCC(=O)O)C(=O)N[C@@H](CO)C(=O)N[C@@H](C)C(=O)NCC(=O)N[C@@H]([C@H](CC)C)C(=O)N[C@@H](CC1=CN=C[N]1[H])C(=O)O

InChI=1S/C25H40N8O10/c1-4-12(2)20(24(41)31-16(25(42)43)7-14-8-27-11-29-14)33-18(35)9-28-21(38)13(3)30-23(40)17(10-34)32-22(39)15(26)5-6-19(36)37/h8,11-13,15-17,20,34H,4-7,9-10,26H2,1-3H3,(H,27,29)(H,28,38)(H,30,40)(H,31,41)(H,32,39)(H,33,35)(H,36,37)(H,42,43)/t12-,13-,15-,16-,17-,20-/m0/s1

InChIKey=NFBYCMWYFUISGO-GZKRCTFISA-N


Peptide identified in thornback ray muscle (Raja clavata) Bacillus subtilis A26 hydrolysate. IC50 value of synthetic peptide was 371.60 uM.



Database reference:
EROP-Moscow: ID E25022