BIOPEP-UWM: Report

ID 9038
Name ACE inhibitor
sequence
SVY

Function:
Inhibitor of Angiotensin-Converting Enzyme (ACE) (EC 3.4.15.1) (MEROPS ID: M02-001)
 
Number of residues
3
Activity code
ah
Activity :
ACE inhibitor
Chemical mass 367.3959 Monoisotopic mass 367.1737
IC50 :
8.13 µM



Bibliographic data:
Authors
Wu J., Aluko R. E., Nakai S.
Title
Structural requirements of angiotensin I-converting enzyme inhibitory activity: quantitative structure-activity relationship study of di- and tripeptides. J. Agric. Food Chem., 54, 732-738, 2006
Year Source
2006 Journal



Additional information:
BIOPEP-UWM database of bioactive peptides


SMILES: N[C@@]([H])(CO)C(=O)N[C@@]([H])(C(C)C)C(=O)N[C@@]([H])(Cc1ccc(O)cc1)C(=O)O

InChI=1S/C17H25N3O6/c1-9(2)14(20-15(23)12(18)8-21)16(24)19-13(17(25)26)7-10-3-5-11(22)6-4-10/h3-6,9,12-14,21-22H,7-8,18H2,1-2H3,(H,19,24)(H,20,23)(H,25,26)/t12-,13-,14-/m0/s1

InChIKey: ODRUTDLAONAVDV-IHRRRGAJSA-N


Information concerning Angiotensin-Converting Enzyme (ACE) is available in MEROPS database of proteolytic enzymes (http://merops.sanger.ac.uk/); ID: M02-001



Database reference:
AHTPDB: ID 1562, 1629

BioPepDB: ID biopep01268

J-GLOBAL: ID 200907071997017328

Nikkaji: ID J982.302F

PubChem: CID 102123472

SATPdb: ID satpdb11953