BIOPEP-UWM: Report

ID 9064
Name ACE inhibitor
sequence
LEK

Function:
Inhibitor of Angiotensin-Converting Enzyme (ACE) (EC 3.4.15.1) (MEROPS ID: M02-001)
 
Number of residues
3
Activity code
ah
Activity :
ACE inhibitor
Chemical mass 388.4579 Monoisotopic mass 388.2314
EC50 :
794.40 µM



Bibliographic data:
Authors
Wu J., Aluko R. E., Nakai S.
Title
Structural requirements of angiotensin I-converting enzyme inhibitory activity: quantitative structure-activity relationship study of di- and tripeptides. J. Agric. Food Chem., 54, 732-738, 2006
Year Source
2006 Journal



Additional information:
BIOPEP-UWM database of bioactive peptides


SMILES: N[C@@]([H])(CC(C)C)C(=O)N[C@@]([H])(CCC(=O)O)C(=O)N[C@@]([H])(CCCCN)C(=O)O

InChI=1S/C17H32N4O6/c1-10(2)9-11(19)15(24)20-12(6-7-14(22)23)16(25)21-13(17(26)27)5-3-4-8-18/h10-13H,3-9,18-19H2,1-2H3,(H,20,24)(H,21,25)(H,22,23)(H,26,27)/t11-,12-,13-/m0/s1

InChIKey: HQUXQAMSWFIRET-AVGNSLFASA-N


Information concerning Angiotensin-Converting Enzyme (ACE) is available in MEROPS database of proteolytic enzymes (http://merops.sanger.ac.uk/); ID: M02-001



Database reference:
AHTPDB: ID 1630, 2856

BioPepDB: ID biopep00747

ChemSpider: ID 9592739

PubChem: CID 11417852

SATPdb: ID satpdb13310