BIOPEP-UWM: Report

ID 9109
Name ACE inhibitor
sequence
LIWKL

Function:
Inhibitor of Angiotensin-Converting Enzyme (ACE) (EC 3.4.15.1) (MEROPS ID: M02-001)
 
Number of residues
5
Activity code
ah
Activity :
ACE inhibitor
Chemical mass 671.8681 Monoisotopic mass 671.4357
IC50 :
0.47 µM



Bibliographic data:
Authors
Ruiz-Giménez P., Salom J. B., Marcos J. F., Valles S., Martinez-Maqueda D., Recio I., Torregrosa G., Alborch E., Manzanares P.
Title
Antihypertensive effect of a bovine lactoferrin pepsin hydrolysate: Identification of novel active peptides. Food Chem., 131, 266-273, 2012
Year Source
2012 Journal



Additional information:
BIOPEP-UWM database of bioactive peptides


SMILES: N[C@@H](CC(C)C)C(=O)N[C@@H]([C@@H](C)CC)C(=O)N[C@@H](Cc1c2ccccc2[nH]c1)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CC(C)C)C(=O)O

InChI=1S/C35H57N7O6/c1-7-22(6)30(42-31(43)25(37)16-20(2)3)34(46)40-28(18-23-19-38-26-13-9-8-12-24(23)26)33(45)39-27(14-10-11-15-36)32(44)41-29(35(47)48)17-21(4)5/h8-9,12-13,19-22,25,27-30,38H,7,10-11,14-18,36-37H2,1-6H3,(H,39,45)(H,40,46)(H,41,44)(H,42,43)(H,47,48)/t22-,25-,27-,28-,29-,30-/m0/s1

InChIKey: DVGVKGVPVPRABU-KHDOVFMSSA-N


Information concerning Angiotensin-Converting Enzyme (ACE) is available in MEROPS database of proteolytic enzymes (http://merops.sanger.ac.uk/); ID: M02-001



Database reference:
AHTPDB: ID 4331, 5522

BioPepDB: ID biopep00793

MBPDB: peptide LIWKL

SATPdb: ID satpdb25760