BIOPEP-UWM: Report

ID 9112
Name ACE inhibitor
sequence
DAQSAPLRVY

Function:
Inhibitor of Angiotensin-Converting Enzyme (ACE) (EC 3.4.15.1) (MEROPS ID: M02-001)
 
Number of residues
10
Activity code
ah
Activity :
ACE inhibitor
Chemical mass 1119.2247 Monoisotopic mass 1118.5702
IC50 :
13.00 µM



Bibliographic data:
Authors
Tavares T., del Mar Contreras M., Amorim M., Pintado M., Recio I., Malcata F. X.
Title
Novel whey-derived peptides with inhibitory effect against angiotensin-converting enzyme: in vitro effect and stability to gastrointestinal enzymes. Peptides, 32, 1013-1019, 2011
Year Source
2011 Journal



Additional information:

BIOPEP-UWM database of bioactive peptides


SMILES: N[C@@]([H])(CC(=O)O)C(=O)N[C@@]([H])(C)C(=O)N[C@@]([H])(CCC(=O)N)C(=O)N[C@@]([H])(CO)C(=O)N[C@@]([H])(C)C(=O)N1[C@@]([H])(CCC1)C(=O)N[C@@]([H])(CC(C)C)C(=O)N[C@@]([H])(CCCNC(=N)N)C(=O)N[C@@]([H])(C(C)C)C(=O)N[C@@]([H])(Cc1ccc(O)cc1)C(=O)O

InChI=1S/C49H78N14O16/c1-23(2)19-32(43(73)58-30(9-7-17-54-49(52)53)42(72)62-38(24(3)4)46(76)60-33(48(78)79)20-27-11-13-28(65)14-12-27)59-45(75)35-10-8-18-63(35)47(77)26(6)56-44(74)34(22-64)61-41(71)31(15-16-36(51)66)57-39(69)25(5)55-40(70)29(50)21-37(67)68/h11-14,23-26,29-35,38,64-65H,7-10,15-22,50H2,1-6H3,(H2,51,66)(H,55,70)(H,56,74)(H,57,69)(H,58,73)(H,59,75)(H,60,76)(H,61,71)(H,62,72)(H,67,68)(H,78,79)(H4,52,53,54)/t25-,26-,29-,30-,31-,32-,33-,34-,35-,38-/m0/s1

InChIKey: OVZGOCMQQXSJSD-UQIDJKEMSA-N


Information concerning Angiotensin-Converting Enzyme (ACE) is available in MEROPS database of proteolytic enzymes (http://merops.sanger.ac.uk/); ID: M02-001



Database reference:
AHTPDB: ID 1299, 2546

BioPepDB: ID biopep00118

MBPDB: Peptide DAQSAPLRVY

SATPdb: ID satpdb28591