BIOPEP-UWM: Report

ID 9773
Name Prolyl endopeptidase inhibitor
sequence
VEIPE

Function:
Inhibitor of Prolyl Endopeptidase (EC 3.4.21.26) (MEROPS ID: S09.001)
 
Number of residues
5
Activity code
am
Activity :
antiamnestic
Chemical mass 585.6454 Monoisotopic mass 585.2999
IC50 :
17.00 µM



Bibliographic data:
Authors
Yanai T., Suzuki Y., Sato M.
Title
Prolyl Endopeptidase Inhibitory Peptides in Wine. Bioscience, Biotechnology, and Biochemistry, 67(2), 380–382, 2003
Year Source
2003 Journal



Additional information:
BIOPEP-UWM database of bioactive peptides


SMILES: N[C@@]([H])(C(C)C)C(=O)N[C@@]([H])(CCC(=O)O)C(=O)N[C@@]([H])([C@]([H])(CC)C)C(=O)N1[C@@]([H])(CCC1)C(=O)N[C@@]([H])(CCC(=O)O)C(=O)O


InChI=1S/C26H43N5O10/c1-5-14(4)21(30-22(36)15(8-10-18(32)33)28-24(38)20(27)13(2)3)25(39)31-12-6-7-17(31)23(37)29-16(26(40)41)9-11-19(34)35/h13-17,20-21H,5-12,27H2,1-4H3,(H,28,38)(H,29,37)(H,30,36)(H,32,33)(H,34,35)(H,40,41)/t14-,15-,16-,17-,20-,21-/m0/s1


InChIKey: NVPOPSZOSXDRSP-KZVLABISSA-N



Database reference:
BRENDA: Ligand Val-Glu-Ile-Pro-Glu

ChemSpider: ID 8364095

J-GLOBAL: ID 200907071043205077

Nikkaji: ID J1.559.065C