BIOPEP-UWM: Report

ID 9917
Name Inhibitor of tripeptidyl peptidase 2
sequence
VA
Function:
Inhibitor of Tripeptidyl peptidase 2 (TPP 2) (EC 3.4.14.10) (MEROPS ID: S08.090)
 
Number of residues
2
Activity code
tpp2
Activity :
inhibitor of tripeptidyl peptidase II
Chemical mass 188.2236 Monoisotopic mass 188.1157
EC50 :
0.00 µM


Bibliographic data:
Authors
Ganellin C. R., Bishop P. B., Bambal R. B., Chan S. M., Law J. K., Marabout B., Luthra P. M., Moore A. N., Peschard O., Bourgeat P., Rose C., Vargas F., Schwartz J. C.
Title
Inhibitors of tripeptidyl peptidase II. 2. Generation of the first novel lead inhibitor of cholecystokinin-8-inactivating peptidase: a strategy for the design of peptidase inhibitors. J. Med. Chem., 43, 664-674, 2000
Year Source
2000 Journal


Additional information:
BIOPEP-UWM database of bioactive peptides


SMILES: N[C@@H](C(C)C)C(=O)N[C@@H](C)C(=O)O

InChI=1S/C8H16N2O3/c1-4(2)6(9)7(11)10-5(3)8(12)13/h4-6H,9H2,1-3H3,(H,10,11)(H,12,13)/t5-,6-/m0/s1

InChIKey: HSRXSKHRSXRCFC-WDSKDSINSA-N


Inhibitor of Dipeptidyl Peptidase IV (EC 3.4.14.5) (MEROPS ID: S09.003) according to the BIOPEP-UWM database of biactive peptides (ID 3172)
Inhibitor of Angiotensin-converting enzyme (EC 3.4.15.1) (MEROPS ID: M02-001) according to the AHTPDB database


Bitter peptide according to the BIOPEP-UWM database of sensory peptides and amino acids, the ChEMBL database


Database reference:
AHTPDB: ID 3848

BIOPEP-UWM database of bioactive peptides: ID 3172

BIOPEP-UWM database of sensory peptides and amino acids: ID 462

BRENDA: Ligand Val-Ala

ChEBI: ID 75008

ChEMBL: ID CHEMBL55523

ChemSpider: ID 5360762

CompTox: ID DTXSID60426328

EPA DSSTox: ID DTXCID40377162

EROP-Moscow: ID E09235

J-GLOBAL: ID 200907035026970731

Nikkaji: ID J149.658A

PubChem: CID 6992637

SATPdb: ID satpdb14267

ZINC: ID ZINC01578617