BIOPEP-UWM: Report

ID 345
Name Bitter peptide
sequence
LVYPFPGPIHN

Function:
Bitter taste
 
Number of residues
11
Activity code
bi
Activity :
bitter
Chemical mass 1253.4440 Monoisotopic mass 1252.6584
EC50 :
0.00 µM



Bibliographic data:
Authors
Kohl S., Behrens M., Dunkel A., Hofmann T., Meyerhof W.
Title
Amino acids and peptides activate at least five members of the human bitter taste receptor family. J. Agric. Food Chem., 61, 53-60
Year Source
2013 Journal



Additional information:
BIOPEP database of sensory peptides and amino acids


SMILES: N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N1[C@H](C(=O)N[C@H](C(=O)N2[C@H](C(=O)NCC(=O)N3[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)O)CC(=O)N)Cc4[nH]cnc4)[C@H](CC)C)CCC3)CCC2)Cc2ccccc2)CCC1)Cc1ccc(cc1)O)C(C)C)CC(C)C

InChI=1S/C62H88N14O14/c1-7-36(6)52(59(86)68-42(29-39-31-65-33-67-39)54(81)71-45(62(89)90)30-49(64)78)73-57(84)47-17-11-23-74(47)50(79)32-66-55(82)46-16-12-24-75(46)60(87)43(27-37-14-9-8-10-15-37)69-56(83)48-18-13-25-76(48)61(88)44(28-38-19-21-40(77)22-20-38)70-58(85)51(35(4)5)72-53(80)41(63)26-34(2)3/h8-10,14-15,19-22,31,33-36,41-48,51-52,77H,7,11-13,16-18,23-30,32,63H2,1-6H3,(H2,64,78)(H,65,67)(H,66,82)(H,68,86)(H,69,83)(H,70,85)(H,71,81)(H,72,80)(H,73,84)(H,89,90)/t36-,41-,42-,43-,44-,45-,46-,47-,48-,51-,52-/m0/s1

InChIKey: GQLLYOVQTZKCLF-LVEINZFUSA-N



Database reference:
BindingDB: ID 50169218

BIOPEP database of bioactive peptides: ID 8681

ChEMBL: ID CHEMBL434535

ChemSpider: ID 23257174

PubChem: ID 44398561