BIOPEP-UWM: Report

ID 40
Name bitter peptide
sequence
YYY

Function:
(Rcaf) 5
 
Number of residues
3
Activity code
bi
Activity :
bitter
Chemical mass 507.5339 Monoisotopic mass 507.1998
EC50 :
0.00 µM



Bibliographic data:
Authors
Ishibashi N., Sadamori K., Yamamoto O., Kanehisa H., Kouge K., Kikuchi E., Okai H., Fukui S.
Title
Bitterness of phenylalanine- and tyrosine-containing peptides. Agric. Biol. Chem., 51, 3309-3313, 1987
Year Source
1987 Journal



Additional information:
BIOPEP database of sensory peptides and amino acids


SMILES: c1cc(ccc1C[C@@H](C(=O)N[C@@H](Cc2ccc(cc2)O)C(=O)N[C@@H](Cc3ccc(cc3)O)C(=O)O)N)O

InChI=1S/C27H29N3O7/c28-22(13-16-1-7-19(31)8-2-16)25(34)29-23(14-17-3-9-20(32)10-4-17)26(35)30-24(27(36)37)15-18-5-11-21(33)12-6-18/h1-12,22-24,31-33H,13-15,28H2,(H,29,34)(H,30,35)(H,36,37)/t22-,23-,24-/m0/s1

InChIKey: RMRFSFXLFWWAJZ-HJOGWXRNSA-N


Angiotensin-converting enzyme (EC 3.4.15.1) (MEROPS ID: XM02-001) inhibitor according to AHTPDB database
Antioxidative peptide according to BIOPEP database of bioactive peptides
Inhibitor of citrulline uptake in yeasts according to ChEMBL database



Database reference:


AHTPDB: ID 4566; 4871; 5480;

BIOPEP database of bioactive peptides: ID 7945;

BRENDA: Ligand Tyr-Tyr-Tyr;

ChEMBL: ID CHEMBL1221566;

ChemSpider: ID 24022629;

PubChem ID: 40520321