BIOPEP-UWM: Report

ID 143
Name Acetylcholinesterase inhibitor
sequence
HRMLLRRYY

Function:
Predicted ligand of Acetylcholinesterase (EC 3.1.1.7) (PDB ID: 4BDT)
 
Number of residues
9
Activity code
ache
Activity :
AChE inhibitor
Chemical mass 1307.5668 Monoisotopic mass 1306.7061
EC50 :
0.00 µM



Bibliographic data:
Authors
Dastan D., Zhiyani R., Fasihi K., Ebadi A.
Title
An arginine-rich peptide inhibits AChE: template-based design, molecular modeling, synthesis and biological evaluation. J. Mol. Model., 28, 86, 2022
Year Source
2022 Journal



Additional information:
BIOPEP-UWM Virtual database


SMILES: N[C@@H](CC1=CN=C[NH]1)C(=O)N[C@@]([H])(CCCNC(=N)N)C(=O)N[C@@]([H])(CCSC)C(=O)N[C@@]([H])(CC(C)C)C(=O)N[C@@]([H])(CC(C)C)C(=O)N[C@@]([H])(CCCNC(=N)N)C(=O)N[C@@]([H])(CCCNC(=N)N)C(=O)N[C@@H](CC1=CC=C(C=C1)O)C(=O)N[C@@H](CC1=CC=C(C=C1)O)C(=O)O

InChI=1S/C59H94N20O12S/c1-32(2)25-44(77-54(88)45(26-33(3)4)76-52(86)43(20-24-92-5)75-49(83)40(9-6-21-68-57(61)62)72-48(82)39(60)29-36-30-67-31-71-36)53(87)74-41(10-7-22-69-58(63)64)50(84)73-42(11-8-23-70-59(65)66)51(85)78-46(27-34-12-16-37(80)17-13-34)55(89)79-47(56(90)91)28-35-14-18-38(81)19-15-35/h12-19,30-33,39-47,80-81H,6-11,20-29,60H2,1-5H3,(H,67,71)(H,72,82)(H,73,84)(H,74,87)(H,75,83)(H,76,86)(H,77,88)(H,78,85)(H,79,89)(H,90,91)(H4,61,62,68)(H4,63,64,69)(H4,65,66,70)/t39-,40-,41-,42-,43-,44-,45-,46-,47-/m0/s1

InChIKey=GADWILQXLSPBKA-CSYZDTNESA-N


Bioactivity predicted using molecular docking



Database reference: