BIOPEP-UWM: Report

ID 257
Name PPARγ antagonist
sequence
IIQGR

Function:
Predicted ligand of PPARγ (PDB ID: 3V9V)
 
Number of residues
5
Activity code
ppar
Activity :
PPARγ antagonist
Chemical mass 585.6949 Monoisotopic mass 585.3588
EC50 :
0.00 µM



Bibliographic data:
Authors
Ruiz-López F. d. J., Espinosa-Rodríguez B. A., Silva-Mares D. A., González-Martínez B. E., López-Cabanillas Lomelí M., Méndez-López L. F. et al.
Title
In silico identification of peptides with PPARγ antagonism in protein hydrolysate from rice (Oryza sativa). Pharmaceuticals, 16, 440, 2023
Year Source
2023 Journal



Additional information:
BIOPEP-UWM Virtual database


SMILES: N[C@@]([H])([C@]([H])(CC)C)C(=O)N[C@@]([H])([C@]([H])(CC)C)C(=O)N[C@@]([H])(CCC(=O)N)C(=O)NCC(=O)N[C@@]([H])(CCCNC(=N)N)C(=O)O

InChI=1S/C25H47N9O7/c1-5-13(3)19(27)22(38)34-20(14(4)6-2)23(39)33-15(9-10-17(26)35)21(37)31-12-18(36)32-16(24(40)41)8-7-11-30-25(28)29/h13-16,19-20H,5-12,27H2,1-4H3,(H2,26,35)(H,31,37)(H,32,36)(H,33,39)(H,34,38)(H,40,41)(H4,28,29,30)/t13-,14-,15-,16-,19-,20-/m0/s1

InChIKey=FSZJEPJJKFNZBS-IGVQRDAMSA-N



Database reference: