BIOPEP-UWM: Report

ID 258
Name PPARγ antagonist
sequence
QPY

Function:
Predicted ligand of PPARγ (PDB ID: 3V9V)
 
Number of residues
3
Activity code
ppar
Activity :
PPARγ antagonist
Chemical mass 406.4319 Monoisotopic mass 406.1846
EC50 :
0.00 µM



Bibliographic data:
Authors
Ruiz-López F. d. J., Espinosa-Rodríguez B. A., Silva-Mares D. A., González-Martínez B. E., López-Cabanillas Lomelí M., Méndez-López L. F. et al.
Title
In silico identification of peptides with PPARγ antagonism in protein hydrolysate from rice (Oryza sativa). Pharmaceuticals, 16, 440, 2023
Year Source
2023 Journal



Additional information:
BIOPEP-UWM Virtual database


SMILES: N[C@@]([H])(CCC(=O)N)C(=O)N1[C@@]([H])(CCC1)C(=O)N[C@@H](CC1=CC=C(C=C1)O)C(=O)O

InChI=1S/C19H26N4O6/c20-13(7-8-16(21)25)18(27)23-9-1-2-15(23)17(26)22-14(19(28)29)10-11-3-5-12(24)6-4-11/h3-6,13-15,24H,1-2,7-10,20H2,(H2,21,25)(H,22,26)(H,28,29)/t13-,14-,15-/m0/s1

InChIKey=DCWNCMRZIZSZBL-KKUMJFAQSA-N



Database reference:
ChEBI: ID 162450

Metabolomics Workbench: ID 81354

PubChem: CID 145455194