BIOPEP-UWM: Report

ID 259
Name PPARγ antagonist
sequence
QSPVF

Function:
Predicted ligand of PPARγ (PDB ID: 3V9V)
 
Number of residues
5
Activity code
ppar
Activity :
PPARγ antagonist
Chemical mass 576.6403 Monoisotopic mass 576.2898
EC50 :
0.00 µM



Bibliographic data:
Authors
Ruiz-López F. d. J., Espinosa-Rodríguez B. A., Silva-Mares D. A., González-Martínez B. E., López-Cabanillas Lomelí M., Méndez-López L. F., Vázquez-Rod
Title
In silico identification of peptides with PPARγ antagonism in protein hydrolysate from rice (Oryza sativa). Pharmaceuticals, 16, 440, 2023
Year Source
2023 Journal



Additional information:
BIOPEP-UWM Virtual database


SMILES: N[C@@]([H])(CCC(=O)N)C(=O)N[C@@]([H])(CO)C(=O)N1[C@@]([H])(CCC1)C(=O)N[C@@]([H])(C(C)C)C(=O)N[C@@H](CC1=CC=C(C=C1))C(=O)O

InChI=1S/C27H40N6O8/c1-15(2)22(25(38)30-18(27(40)41)13-16-7-4-3-5-8-16)32-24(37)20-9-6-12-33(20)26(39)19(14-34)31-23(36)17(28)10-11-21(29)35/h3-5,7-8,15,17-20,22,34H,6,9-14,28H2,1-2H3,(H2,29,35)(H,30,38)(H,31,36)(H,32,37)(H,40,41)/t17-,18-,19-,20-,22-/m0/s1

InChIKey=JSEQEJRNSOYFDN-HVAMYJMISA-N



Database reference: