BIOPEP-UWM: Report

ID 601
Name ACE inhibitor
sequence
HPF

Function:
Predicted inhibitor of Angiotensin-Converting Enzyme (ACE) (EC 3.4.15.1) (MEROPS ID: M02-001)
 
Number of residues
3
Activity code
ah
Activity :
ACE inhibitor
Chemical mass 399.4426 Monoisotopic mass 399.1901
EC50 :
0.00 µM



Bibliographic data:
Authors
Gu J., Yue S., Yang X., Lu Z., Wang Z., Wei X., Zhou L., Zhao Z., Shi Z., Zhao Z.
Title
Unlocking novel angiotensin-converting enzyme inhibitory peptides from Nili Ravi buffalo milk β-casein: A synergistic strategy combining targeted hydrolysis, 3D-QSAR modeling, and mechanistic insights. Food Biosci., 71, 107346, 2025
Year Source
2025 Journal



Additional information:
BIOPEP-UWM Virtual database


SMILES: N[C@@H](CC1=CN=C[NH]1)C(=O)N1[C@@]([H])(CCC1)C(=O)N[C@@H](CC1=CC=C(C=C1))C(=O)O

InChI=1S/C20H25N5O4/c21-15(10-14-11-22-12-23-14)19(27)25-8-4-7-17(25)18(26)24-16(20(28)29)9-13-5-2-1-3-6-13/h1-3,5-6,11-12,15-17H,4,7-10,21H2,(H,22,23)(H,24,26)(H,28,29)/t15-,16-,17-/m0/s1

InChIKey=PBVQWNDMFFCPIZ-ULQDDVLXSA-N


Activity predicted using QSAR


Angiotensin II receptor ligand according to the BindingDB database; the ChEMBL database



Database reference:
BindingDB: ID BDBM50208103

BRENDA: Ligand His-Pro-Phe

CAS: Registry No 31025-44-2

ChEBI: ID CHEBI:157911

ChEMBL: ID CHEMBL385998

EPA DSSTox: ID DTXSID80437698

J-GLOBAL: ID 200907063797982310

Metabolomics Workbench: ID 82549

Nikkaji: ID J2.719.892I

PubChem: CID 10272250

SureChEMBL: ID SCHEMBL29649768

UniChem: ID 257302

Wikidata: ID Q76415388