BIOPEP-UWM: Report

ID 82
Name ACE inhibitor
sequence
YLLDLLPAAASHR

Function:
Predicted inhibitor of Angiotensin-Converting Enzyme (ACE) (EC 3.4.15.1) (MEROPS ID: M02-001) (PDB ID: 1O86)
 
Number of residues
13
Activity code
ah
Activity :
ACE inhibitor
Chemical mass 1439.6534 Monoisotopic mass 1438.7908
EC50 :
0.00 µM



Bibliographic data:
Authors
Marcet I., Delgado J., Díaz N., Rendueles M., Díaz M.
Title
Peptides recovery from egg yolk lipovitellins by ultrafiltration and their in silico bioactivity analysis. Food Chem., 379, 132145, 2022
Year Source
2022 Journal



Additional information:
BIOPEP-UWM Virtual database


SMILES: N[C@@H](CC1=CC=C(C=C1)O)C(=O)N[C@@]([H])(CC(C)C)C(=O)N[C@@]([H])(CC(C)C)C(=O)N[C@@]([H])(CC(=O)O)C(=O)N[C@@]([H])(CC(C)C)C(=O)N[C@@]([H])(CC(C)C)C(=O)N1[C@@]([H])(CCC1)C(=O)N[C@@]([H])(C)C(=O)N[C@@]([H])(C)C(=O)N[C@@]([H])(C)C(=O)N[C@@]([H])(CO)C(=O)N[C@@H](CC1=CN=C[NH]1)C(=O)N[C@@]([H])(CCCNC(=N)N)C(=O)O

InChI=1S/C66H106N18O18/c1-32(2)22-44(77-56(92)42(67)26-39-16-18-41(86)19-17-39)57(93)78-45(23-33(3)4)58(94)81-48(28-52(87)88)61(97)79-46(24-34(5)6)59(95)82-49(25-35(7)8)64(100)84-21-13-15-51(84)63(99)75-37(10)54(90)73-36(9)53(89)74-38(11)55(91)83-50(30-85)62(98)80-47(27-40-29-70-31-72-40)60(96)76-43(65(101)102)14-12-20-71-66(68)69/h16-19,29,31-38,42-51,85-86H,12-15,20-28,30,67H2,1-11H3,(H,70,72)(H,73,90)(H,74,89)(H,75,99)(H,76,96)(H,77,92)(H,78,93)(H,79,97)(H,80,98)(H,81,94)(H,82,95)(H,83,91)(H,87,88)(H,101,102)(H4,68,69,71)/t36-,37-,38-,42-,43-,44-,45-,46-,47-,48-,49-,50-,51-/m0/s1

InChIKey=ZSIOMTAWGFFBDF-KIMVUHIKSA-N


Bioactivity predicted by molecular docking




Database reference: